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Publication Year

  • 2019
  • 2018
  • 2017
  • 2016

Author

  • Sergio Dall'Angelo
2019

Enzymatic radiosynthesis of a 18F-Glu-Ureido-Lys ligand for the prostate-specific membrane antigen (PSMA)

Lowe, P. T., Dall'Angelo, S., Fleming, I. N., Piras, M., Zanda, M. & O'Hagan, D., 2019, In : Organic & Biomolecular Chemistry. 17, 6, p. 1480-1486 7 p.

Research output: Contribution to journalArticle

Open Access
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4 Citations (Scopus)
3 Downloads (Pure)

The Trifluoromethyl Group as a Bioisosteric Replacement of the Aliphatic Nitro Group in CB1 Receptor Positive Allosteric Modulators (PAMs)

Tseng, C-C., Baillie, G., Donvito, G., Mustafa, M. A., Juola, S. E., Zanato, C., Massarenti, C., Dall'angelo, S., Harrison, W. T. A., Lichtman, A. H., Ross, R. A., Zanda, M. & Greig, I. R., 2019, In : Journal of Medicinal Chemistry. 62, 10, p. 5049-5062 14 p.

Research output: Contribution to journalArticle

Open Access
File
7 Citations (Scopus)
3 Downloads (Pure)
2018
Open Access
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10 Citations (Scopus)
9 Downloads (Pure)

Enzymatic Fluorination of Biotin and Tetrazine Conjugates for Pretargeting Approaches to Positron Emission Tomography Imaging

Lowe, P. T., Dall'angelo, S., Devine, A., Zanda, M. & O'Hagan, D., 17 Sep 2018, In : ChemBioChem. 19, 18, p. 1969-1978 10 p.

Research output: Contribution to journalArticle

Open Access
File
7 Citations (Scopus)
3 Downloads (Pure)

Preclinical Evaluation of [18F]LCATD as a PET Tracer to Study Drug-Drug Interactions Caused by Inhibition of Hepatic Transporters

Testa, A., Dall'Angelo, S., Mingarelli, M., Augello, A., Schweiger, L., Welch, A., Elmore, C. S., Dawson, D., Sharma, P. & Zanda, M., 30 Jul 2018, In : Contrast Media & Molecular Imaging. 2018, 10 p., 3064751.

Research output: Contribution to journalArticle

Open Access
File
10 Downloads (Pure)
2017

A New Class of Fluorinated A2A Adenosine Receptor Agonist with Application to Last-Step Enzymatic 18F Fluorination for PET Imaging

Lowe, P. T., Dall'Angello, S., Mulder-Krieger, T., Ijzerman, A. P., Zanda, M. & O'Hagan, D., 2 Nov 2017, In : ChemBioChem. 18, 21, p. 2156-2164 9 p.

Research output: Contribution to journalArticle

Open Access
File
7 Citations (Scopus)
9 Downloads (Pure)

Design, synthesis, in vitro characterization and preliminary imaging studies on fluorinated bile acid derivatives as PET tracers to study hepatic transporters

Testa, A., Dall'Angelo, S., Mingarelli, M., Augello, A., Schweiger, L., Welch, A. E., Elmore, C. S., Sharma, P. & Zanda, M., 1 Feb 2017, In : Bioorganic & Medicinal Chemistry. 25, 3, p. 963-976 14 p.

Research output: Contribution to journalArticle

Open Access
File
11 Citations (Scopus)
9 Downloads (Pure)

High Affinity “Click” RGD Peptidomimetics as Radiolabeled Probes for Imaging αvβ3 Integrin

Piras, M., Testa, A., Fleming, I. N., Dall'Angelo, S., Andriu, A., Menta, S., Mori, M., Brown, G. D., Forster, D., Williams, K. J. & Zanda, M., 20 Jul 2017, In : ChemMedChem. 12, 14, p. 1142-1151 10 p.

Research output: Contribution to journalArticle

Open Access
File
6 Citations (Scopus)
10 Downloads (Pure)

Synthesis, radio-synthesis and in vitro evaluation of terminally fluorinated derivatives of HU-210 and HU-211 as novel candidate PET tracers

Zanato, C., Pelagalli, A., Marwick, K. F. M., Piras, M., Dall'Angelo, S., Spinaci, A., Pertwee, R. G., Wyllie, D. J. A., Hardingham, G. E. & Zanda, M., 2017, In : Organic & Biomolecular Chemistry. 15, 9, p. 2086-2096 11 p.

Research output: Contribution to journalArticle

Open Access
File
3 Citations (Scopus)
9 Downloads (Pure)

Synthesis and hyperpolarisation of eNOS substrates for quantification of NO production by (1)H NMR spectroscopy

Fernandez Diaz-Rullo, F., Zamberlan, F., Mewis, R. E., Fekete, M., Broche, L., Cheyne, L. A., Dall'Angelo, S., Duckett, S. B., Dawson, D. & Zanda, M., 15 May 2017, In : Bioorganic & Medicinal Chemistry. 25, 10, p. 2730-2742 13 p.

Research output: Contribution to journalArticle

Open Access
File
4 Citations (Scopus)
6 Downloads (Pure)

Synthesis and radio-synthesis of prospective 2-nitroimidazole hypoxia PET tracers via thiazolidine ligation with 5-fluorodeoxyribose (FDR)

Musolino, M., Dall'angelo, S. & Zanda, M., 2017, In : SynOpen. 1, 1, p. 173-179 7 p.

Research output: Contribution to journalArticle

Open Access
File
6 Downloads (Pure)

Synthesis and Superpotent Anticancer Activity of Tubulysins Carrying Non-hydrolysable N-Substituents on Tubuvaline

Sani, M., Lazzari, P., Folini, M., Spiga, M., Zuco, V., De Cesare, M., Manca, I., Dall'Angelo, S., Frigerio, M., Usai, I., Testa, A., Zaffaroni, N. & Zanda, M., 27 Apr 2017, In : Chemistry : a European Journal. 23, 24, p. 5842-5850 9 p.

Research output: Contribution to journalArticle

Open Access
File
5 Citations (Scopus)
8 Downloads (Pure)
2016

Last-step enzymatic [18F]-fluorination of cysteine-tethered RGD peptides using modified Barbas linkers

Zhang, Q., Dall'Angelo, S., Fleming, I. N., Schweiger, L. F., Zanda, M. & O'Hagan, D., 25 Jul 2016, In : Chemistry : a European Journal. 22, 31, p. 10998-11004 7 p.

Research output: Contribution to journalArticle

Open Access
File
17 Citations (Scopus)
7 Downloads (Pure)

NGR Tumor-Homing Peptides: Structural Requirements for Effective APN (CD13) Targeting

Graziadio, A., Zanda, M., Frau, S., Fleming, I. N., Musolino, M., Dall'Angelo, S., Baldassarre, M. & Piras, M., 18 May 2016, In : Bioconjugate Chemistry. 27, 5, p. 1332-1340 9 p.

Research output: Contribution to journalArticle

Open Access
File
17 Citations (Scopus)
7 Downloads (Pure)